Adding a Lysine Mimic in the Design of Potent Inhibitors of Histone Lysine Methyltransferases-Reference-Cited by-同舟云学术

登录注册会员服务联系我们

Adding a Lysine Mimic in the Design of Potent Inhibitors of Histone Lysine Methyltransferases

Published:2010-07 Issue:1 Volume:400 Page:1-7
ISSN:0022-2836
Container-title:Journal of Molecular Biology
language:en
Short-container-title:Journal of Molecular Biology

Author:

Chang Yanqi,Ganesh Thota,Horton John R.,Spannhoff Astrid,Liu Jin,Sun Aiming,Zhang Xing,Bedford Mark T.,Shinkai Yoichi,Snyder James P.,Cheng Xiaodong

Publisher

Elsevier BV

Subject

Molecular Biology,Structural Biology

Reference18 articles.

1. Chemical probes for histone-modifying enzymes;Cole;Nat. Chem. Biol.,2008

2. Protein methyltransferases as a target class for drug discovery;Copeland;Nat. Rev., Drug Discov.,2009

3. Reversal of H3K9me2 by a small-molecule inhibitor for the G9a histone methyltransferase;Kubicek;Mol. Cell,2007

4. Structural basis for G9a-like protein lysine methyltransferase inhibition by BIX-01294;Chang;Nat. Struct. Mol. Biol.,2009

5. Discovery of a 2,4-diamino-7-aminoalkoxyquinazoline as a potent and selective inhibitor of histone lysine methyltransferase G9a;Liu;J. Med. Chem.,2009

Cited by 103 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Discovery of a Highly Potent Lysine Methyltransferases G9a/NSD2 Dual Inhibitor to Treat Solid Tumors;Journal of Medicinal Chemistry;2024-07-15

2. Role of dopamine in the pathophysiology of Parkinson’s disease;Translational Neurodegeneration;2023-09-18

3. Protein Lysine Methyltransferases Inhibitors;Current Medicinal Chemistry;2023-08

4. Structure-Based Design and Characterization of the Highly Potent and Selective Covalent Inhibitors Targeting the Lysine Methyltransferases G9a/GLP;Journal of Medicinal Chemistry;2023-06-02

5. Integration of ligand and structure-based pharmacophore screening for the identification of novel natural leads against Euchromatic histone lysine methyltransferase 2 (EHMT2/G9a);Journal of Biomolecular Structure and Dynamics;2023-05-22

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号京ICP备18003416号-3