Engineering inhibitors highly selective for the S1 sites of Ser190 trypsin-like serine protease drug targets-Reference-Cited by-同舟云学术

Engineering inhibitors highly selective for the S1 sites of Ser190 trypsin-like serine protease drug targets

Published:2001-11 Issue:11 Volume:8 Page:1107-1121
ISSN:1074-5521
Container-title:Chemistry & Biology
language:en
Short-container-title:Chemistry & Biology

Author:

Katz Bradley A,Sprengeler Paul A,Luong Christine,Verner Erik,Elrod Kyle,Kirtley Matt,Janc James,Spencer Jeffrey R,Breitenbucher J.Guy,Hui Hon,McGee Danny,Allen Darin,Martelli Arnold,Mackman Richard L

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,General Medicine,Biochemistry

Reference29 articles.

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3. Selective inhibition of urokinase by substituted phenylguanidines: quantitative structure–activity relationship analyses;Yang;J. Med. Chem.,1990

4. Plasminogen activators, tissue degradation, and cancer;Dano;Adv. Cancer Res.,1985

5. The urokinase-type plasminogen activator system in cancer metastasis: A review;Andreasen;Int. J. Cancer,1997

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