Plasmodium falciparum subtilisin-like protease 1: discovery of potent difluorostatone-based inhibitors-Reference-Cited by-同舟云学术

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Plasmodium falciparum subtilisin-like protease 1: discovery of potent difluorostatone-based inhibitors

Published:2015 Issue:29 Volume:5 Page:22431-22448
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Giovani Simone¹²³⁴⁵,Penzo Maria⁶⁷⁸⁹,Butini Stefania¹²³⁴⁵,Brindisi Margherita¹²³⁴⁵,Gemma Sandra¹²³⁴⁵,Novellino Ettore¹²³⁴¹⁰,Campiani Giuseppe¹²³⁴⁵,Blackman Michael J.⁶⁷⁸⁹,Brogi Simone¹²³⁴⁵

Affiliation:

1. European Research Centre for Drug Discovery and Development (NatSynDrugs)

2. University of Siena

3. Siena

4. Italy

5. Dept. Biotechnology

6. Division of Parasitology

7. MRC National Institute for Medical Research

8. London

9. UK

10. Dip. di Farmacia

Abstract

We here describe the development of potent inhibitors of the malaria parasite enzyme subtilisin-like protease 1 (PfSUB1).

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA01170A

Reference33 articles.

1. WHO World Malaria Report 2013, http://www.who.int/malaria/publications/world_malaria_report_2012/en/, access date 27/10/2014, 08/04/2013)

2. Emergence of artemisinin-resistant malaria on the western border of Thailand: a longitudinal study

3. Multiple populations of artemisinin-resistant Plasmodium falciparum in Cambodia

4. Spread of Artemisinin Resistance in Plasmodium falciparum Malaria

5. If Artemisinin Drugs Fail, What's Plan B?

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