Subtilisin-like Serine Protease 1 (SUB1) as an Emerging Antimalarial Drug Target: Current Achievements in Inhibitor Discovery-Reference-Cited by-同舟云学术

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Subtilisin-like Serine Protease 1 (SUB1) as an Emerging Antimalarial Drug Target: Current Achievements in Inhibitor Discovery

Published:2022-09-22 Issue:19 Volume:65 Page:12535-12545
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lidumniece Elina¹,Withers-Martinez Chrislaine²,Hackett Fiona²,Blackman Michael J.²³^ORCID,Jirgensons Aigars¹^ORCID

Affiliation:

1. Latvian Institute of Organic Synthesis, Riga LV-1006, Latvia

2. Malaria Biochemistry Laboratory, The Francis Crick Institute, London NW1 1AT, United Kingdom

3. Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine, London WC1E 7HT, United Kingdom

Funder

Medical Research Council

Wellcome Trust

Latvijas Zinatnes Padome

Cancer Research UK

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c01093

Reference36 articles.

1. Dihydrofolate reductase and antifolate resistance in malaria

2. Resistance to Artemisinin Combination Therapies (ACTs): Do Not Forget the Partner Drug!

3. Maturation and Specificity of Plasmodium falciparum Subtilisin-like Protease-1, a Malaria Merozoite Subtilisin-like Serine Protease

4. A multistage antimalarial targets the plasmepsins IX and X essential for invasion and egress

5. Malaria Parasite cGMP-dependent Protein Kinase Regulates Blood Stage Merozoite Secretory Organelle Discharge and Egress

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1. Discovery of novel 4-trifluoromethyl-2-anilinoquinoline derivatives as potential anti-cancer agents targeting SGK1;Molecular Diversity;2024-08-09

2. Peptidic Boronic Acid Plasmodium falciparum SUB1 Inhibitors with Improved Selectivity over Human Proteasome;Journal of Medicinal Chemistry;2024-07-25

3. Aryl amino acetamides prevent Plasmodium falciparum ring development via targeting the lipid-transfer protein PfSTART1;Nature Communications;2024-06-18

4. Insights from structure-activity relationships and the binding mode of peptidic α-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1;European Journal of Medicinal Chemistry;2024-04

5. Aryl amino acetamides prevent the development ofPlasmodium falciparumrings via inhibition of the lipid transfer protein PfSTART1;2023-11-04

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