Insights from structure-activity relationships and the binding mode of peptidic α-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1-Reference-Cited by-同舟云学术

Insights from structure-activity relationships and the binding mode of peptidic α-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1

Published:2024-04 Issue: Volume:269 Page:116308
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Legru Alice,Batista Fernando A.,Puszko Anna K.,Bouillon Anthony,Maurel Manon,Martinez Mariano,Ejjoummany Abdelaziz,Ortega Varga Laura,Adler Pauline,Méchaly Ariel,Hadjadj Margot,Sosnowski Piotr,Hopfgartner Gérard,Alzari Pedro M.,Blondel Arnaud,Haouz Ahmed,Barale Jean-Christophe,Hernandez Jean-François^ORCID

Funder

Institut Carnot Chimie Balard Cirimat

French National Research Agency

Horizon 2020

Institut Pasteur

EU Framework Programme for Research and Innovation Marie Skłodowska-Curie Actions

Publisher

Elsevier BV

Reference57 articles.

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3. Emergence and clonal expansion of in vitro artemisinin-resistant Plasmodium falciparum kelch13 R561H mutant parasites in Rwanda;Uwimama;Nat. Med.,2020

4. Evidence of artemisinin-resistant malaria in Africa;Balikagala;N. Engl. J. Med.,2021

5. Artemisinin and multidrug-resistant Plasmodium falciparum - a threat for malaria control and elimination;Dhorda;Curr. Op. Inf. Dis.,2021

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