The facile synthesis of 1-benzoazepine derivatives via gold-catalyzed regioselective cycloisomerization reactions of N-(o-alkynylaryl)-N-vinyl sulfonamides-Reference-Cited by-同舟云学术

The facile synthesis of 1-benzoazepine derivatives via gold-catalyzed regioselective cycloisomerization reactions of N-(o-alkynylaryl)-N-vinyl sulfonamides

Published:2016 Issue:26 Volume:52 Page:4824-4827
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Undeela Sridhar¹²³⁴,Ravikumar Gurram¹²³⁴,Nanubolu Jagadeesh Babu⁵²³⁴,Singarapu Kiran Kumar⁶²³⁴,Menon Rajeev S.¹²³⁴⁷

Affiliation:

1. Medicinal Chemistry and Pharmacology Division

2. CSIR-Indian Institute of Chemical Technology

3. Hyderabad

4. India

5. Centre for X-ray Crystallography

6. Centre for Nuclear Magnetic Resonance

7. Department of Chemistry

Abstract

Gold-catalyzed, regioselective cycloisomerization of N-(o-alkynylaryl)-N-vinyl sulfonamides afforded high yields of 2-sulfonylmethyl-1-benzoazepine derivatives.

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2016/CC/C6CC01061J

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3. Synthesis of N,N′-disubstituted 3-aminobenzo[c] and [d]azepin-2-ones as potent and specific farnesyl transferase inhibitors

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