Discovery of a New-Generation S-Adenosylmethionine-Noncompetitive Covalent Inhibitor Targeting the Lysine Methyltransferase Enhancer of Zeste Homologue 2

Author:

Zhang Yi1,Yang Hong23,Li Bingbing1,Li Jiayi45,Li Huaxuan1,Shi Qiongyu2,Li Bang1,Wang Zekun34,Zheng Jiahong1,Zhang Ying246,Dong Hui1,Huang Xun245,Wang Yuanxiang1ORCID

Affiliation:

1. Balance-Based Drug Discovery Laboratory, School of Pharmaceutical Sciences, Sun Yat-Sen University, Guangzhou 510006, China

2. Lingang Laboratory, Shanghai 200031, China

3. Division of Antitumor Pharmacology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica (SIMM), Chinese Academy of Sciences, Shanghai 201203, China

4. University of Chinese Academy of Sciences, Beijing 100049, China

5. School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou 310024, China

6. School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China

Funder

Shanghai Municipal Health and Family Planning Commission

Science and Technology Commission of Shanghai Municipality

National Natural Science Foundation of China

State Key Laboratory of new Drug development

Guangzhou Basic and Applied Basic Research Foundation

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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