Highly Selective Phosphatidylinositol 4-Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action

Author:

Mejdrová Ivana1,Chalupská Dominika1,Kögler Martin1,Šála Michal1,Plačková Pavla1,Baumlová Adriana1,Hřebabecký Hubert1,Procházková Eliška1,Dejmek Milan1,Guillon Rémi1,Strunin Dmytro1,Weber Jan1,Lee Gary2,Birkus Gabriel2,Mertlíková-Kaiserová Helena1,Boura Evzen1,Nencka Radim1

Affiliation:

1. Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic, v.v.i., Gilead Sciences & IOCB Research Centre, Flemingovo nám. 2, 166 10 Prague 6, Czech Republic

2. Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States

Funder

Ministry of Education, Youth and Sports

Czech Science Foundation

Akademie ved Ceské Republiky

European Commission Directorate-General for Research and Innovation

Gilead Sciences

Seventh Framework Programme

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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