Exploring positions 6 and 7 of a quinazoline-based scaffold leads to changes in selectivity and potency towards RIPK2/3 kinases

Author:

Misehe Mbilo,Matoušová Marika,Dvořáková Alexandra,Hercík Kamil,Škach Kryštof,Chalupská Dominika,Dejmek Milan,Šála Michal,Hájek Miroslav,Boura Evzen,Mertlíková-Kaiserová Helena,Nencka RadimORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference55 articles.

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2. Activation of necroptosis in multiple sclerosis;Ofengeim;Cell Rep.,2015

3. RIP1/RIP3-regulated necroptosis as a target for multifaceted disease therapy;Liu;Int. J. Mol. Med.,2019

4. RIPK2 as a new therapeutic target in inflammatory bowel diseases;Honjo;Front. Pharmacol.,2021

5. Targeting rip kinases in chronic inflammatory disease;Speir;Biomolecules,2021

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