Design, synthesis and evaluation of novel thieno[2,3d]pyrimidine derivatives as potent and specific RIPK2 inhibitors

Author:

Misehe MbiloORCID,Šála Michal,Matoušová MarikaORCID,Hercík Kamil,Kocek HugoORCID,Chalupská Dominika,Chaloupecká Ema,Hájek MiroslavORCID,Boura Evzen,Mertlíková-Kaiserová Helena,Nencka RadimORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference38 articles.

1. Receptor-interacting protein (RIP) kinase family;Zhang;Cellular & Molecular Immunology,2010

2. RIPK protein kinase family: Atypical lives of typical kinases;Cuny;Seminars in Cell & Developmental Biology,2021

3. Function of Nod-like receptors in microbial recognition and host defense;Franchi;Immunological Reviews,2009

4. Essential role of Rip2 in the modulation of innate and adaptive immunity triggered by Nod1 and Nod2 ligands;Magalhaes;European Journal of Immunology,2011

5. NOD Signaling and Cell Death;Heim;Frontiers in Cell and Development Biology,2019

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