In Vitro and In Silico Analysis of the Residence Time of Serotonin 5-HT<sub>7</sub> Receptor Ligands with Arylpiperazine Structure: A Structure–Kinetics Relationship Study-Reference-Cited by-同舟云学术

In Vitro and In Silico Analysis of the Residence Time of Serotonin 5-HT₇ Receptor Ligands with Arylpiperazine Structure: A Structure–Kinetics Relationship Study

Published:2022-01-31 Issue:4 Volume:13 Page:497-509
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Penna Eduardo¹²,Niso Mauro³,Podlewska Sabina⁴^ORCID,Volpicelli Floriana⁵,Crispino Marianna¹,Perrone-Capano Carla⁵⁶,Bojarski Andrzej J.⁴^ORCID,Lacivita Enza³^ORCID,Leopoldo Marcello³^ORCID

Affiliation:

1. Department of Biology, University of Naples Federico II, via Cintia 26, 80126 Naples, Italy

2. Biofordrug srl, via Dante 99, 70019 Triggiano (Bari), Italy

3. Dipartimento di Farmacia-Scienze del Farmaco, Università degli Studi di Bari Aldo Moro, via Orabona 4, 70125 Bari, Italy

4. Maj Institute of Pharmacology, Polish Academy of Sciences, 12 Smętna Street, 31-343 Kraków, Poland

5. Department of Pharmacy, School of Medicine and Surgery, University of Naples Federico II, via Domenico Montesano 49, 80131 Naples, Italy

6. Institute of Genetics and Biophysics “Adriano Buzzati Traverso”, National Research Council (CNR), via Pietro Castellino 111, 80131 Naples, Italy

Funder

Ministero dell?Istruzione, dell?Universit? e della Ricerca

Universita degli Studi di Bari Aldo Moro

Regione Campania

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.1c00710

Reference61 articles.

1. Drug-Target Residence Time-A Case for G Protein-Coupled Receptors

2. The drug–target residence time model: a 10-year retrospective

3. Extrapyramidal side effects of antipsychotics are linked to their association kinetics at dopamine D2 receptors

4. In vivo Target Residence Time and Kinetic Selectivity: The Association Rate Constant as Determinant

5. Ligand Residence Time at G-protein–Coupled Receptors—Why We Should Take Our Time To Study It

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