Drug-Target Residence Time-A Case for G Protein-Coupled Receptors-Reference-Cited by-同舟云学术

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Drug-Target Residence Time-A Case for G Protein-Coupled Receptors

Published:2014-02-18 Issue:4 Volume:34 Page:856-892
ISSN:0198-6325
Container-title:Medicinal Research Reviews
language:en
Short-container-title:Med. Res. Rev.

Author:

Guo Dong¹,Hillger Julia M.¹,IJzerman Adriaan P.¹,Heitman Laura H.¹

Affiliation:

1. Division of Medicinal Chemistry; Leiden Academic Centre for Drug Research; Leiden University; P.O. Box 9502 2300 RA Leiden the Netherlands

Publisher

Wiley

Subject

Drug Discovery,Pharmacology,Molecular Medicine

Reference182 articles.

1. Drug-target residence time and its implications for lead optimization;Copeland;Nat Rev Drug Discov,2006

2. Can binding kinetics translate to a clinically differentiated drug? From theory to practice;Swinney;Lett Drug Des Discov,2006

3. Biochemical mechanisms of new molecular entities (NMEs) approved by United States FDA during 2001-2004: Mechanisms leading to optimal efficacy and safety;Swinney;Curr Top Med Chem,2006

4. How were new medicines discovered;Swinney;Nat Rev Drug Discov,2011

5. Biochemical mechanisms of drug action: What does it take for success?;Swinney;Nat Rev Drug Discov,2004

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