Stereoselective Preparation of a Cyclopentane-Based NK1 Receptor Antagonist Bearing an Unsymmetrically Substituted Sec−Sec Ether
Author:
Affiliation:
1. Department of Process Research, Merck & Company, Incorporated, P.O. Box 2000, Rahway, New Jersey 07065
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/jo061268x
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1. The tachykinin NK1 receptor. Part II: Distribution and pathophysiological roles
2. Discovery of the antidepressant and anti-emetic efficacy of substance P receptor (NK1) antagonists
3. Neurokinin receptor antagonists
4. A Potent Nonpeptide Antagonist of the Substance P (NK 1 ) Receptor
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