A General Method for Acylation of Indoles at the 3-Position with Acyl Chlorides in the Presence of Dialkylaluminum Chloride-Reference-Cited by-同舟云学术

A General Method for Acylation of Indoles at the 3-Position with Acyl Chlorides in the Presence of Dialkylaluminum Chloride

Published:2000-04-27 Issue:10 Volume:2 Page:1485-1487
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Okauchi Tatsuo¹,Itonaga Masaaki¹,Minami Toru¹,Owa Takashi¹,Kitoh Kyosuke¹,Yoshino Hiroshi¹

Affiliation:

1. Department of Applied Chemistry, Kyushu Institute of Technology, 1-1, Sensuicho, Tobata, Kitakyushu, 804-8550, Japan and Tsukuba Research Laboratories, Eisai Company, Ltd., 5-1-3, Tokodai, Tsukuba, 300-2635, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ol005841p

Reference8 articles.

1. Sundberg, R. J.Indoles; Academic Press: New York, 1996; p 113. (b) Pindur, U.; Pfeuffer, L.; Flo, C.Chem.Ztg.1986,110, 307. (c) Engel, R.Chem. Rev.1977,77, 349.

2. N-(Acyloxyalkyl)pyridinium Salts as Soluble Prodrugs of a Potent Platelet Activating Factor Antagonist

3. The Use of Lewis Acid in the Reaction of Zinc Salts of Indoles and Acyl Chloride

4. Entry into 6-Methoxy-D(+)-tryptophans. Stereospecific Synthesis of 1-Benzenesulfonyl-6-methoxy-D(+)-tryptophan Ethyl Ester

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