Rapid Covalent-Probe Discovery by Electrophile-Fragment Screening

Author:

Resnick Efrat,Bradley Anthony12,Gan Jinrui,Douangamath Alice2,Krojer Tobias,Sethi Ritika34,Geurink Paul P.5,Aimon Anthony12,Amitai Gabriel,Bellini Dom6,Bennett James,Fairhead Michael,Fedorov Oleg,Gabizon Ronen,Gan Jin5,Guo Jingxu7,Plotnikov Alexander,Reznik Nava,Ruda Gian Filippo,Díaz-Sáez Laura,Straub Verena M.,Szommer Tamas,Velupillai Srikannathasan,Zaidman Daniel,Zhang Yanling,Coker Alun R.7,Dowson Christopher G.6,Barr Haim M.,Wang ChuORCID,Huber Kilian V.M.ORCID,Brennan Paul E.68ORCID,Ovaa Huib5ORCID,von Delft Frank29,London NirORCID

Affiliation:

1. Department of Chemistry, Chemistry Research Laboratory, 12 Mansfield Road, Oxford OX1 3TA, U.K.

2. Diamond Light Source Ltd., Harwell Science and Innovation Campus, Didcot OX11 0QX, U.K.

3. Structural Biology Research Center, VIB, Brussels, Belgium

4. Structural Biology Brussels, Vrije Universiteit Brussel, Brussels, Belgium

5. Oncode Institute and Department of Cell and Chemical Biology, Leiden University Medical Center, Einthovenweg 20, 2333 ZC Leiden, The Netherlands

6. School of Life Sciences, University of Warwick, Coventry, U.K.

7. Division of Medicine, University College London, Gower Street, London WC1E 6BT, U.K.

8. Alzheimer’s Research UK Oxford Drug Discovery Institute, University of Oxford, NDMRB, Roosevelt Drive, Oxford OX3 7FZ, U.K.

9. Department of Biochemistry, University of Johannesburg, Auckland Park 2006, South Africa

Funder

Israel Science Foundation

Ministry of Science and Technology, Israel

Ontario Genomics Institute

Wellcome Trust

Israel Cancer Research Fund

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

Innovative Medicines Initiative

Rising Tide Foundation

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

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