Efficient Ligand Discovery Using Sulfur(VI) Fluoride Reactive Fragments-Reference-Cited by-同舟云学术

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Efficient Ligand Discovery Using Sulfur(VI) Fluoride Reactive Fragments

Published:2023-04-21 Issue:9 Volume:18 Page:1926-1937
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Aatkar Arron¹²,Vuorinen Aini¹³,Longfield Oliver E.¹²,Gilbert Katharine¹²,Peltier-Heap Rachel⁴,Wagner Craig D.⁴,Zappacosta Francesca⁴,Rittinger Katrin³^ORCID,Chung Chun-wa¹^ORCID,House David¹³^ORCID,Tomkinson Nicholas C. O.²^ORCID,Bush Jacob T.¹³^ORCID

Affiliation:

1. GSK, Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K.

2. Department of Pure and Applied Chemistry, University of Strathclyde, 295 Cathedral Street, Glasgow G1 1XL, U.K.

3. The Francis Crick Institute, London NW1 1AT, U.K.

4. GSK, South Collegeville Road, Collegeville, Pennsylvania 19426, United States

Funder

Engineering and Physical Sciences Research Council

Medical Research Council

Wellcome Trust

Cancer Research UK

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.3c00034

Reference49 articles.

1. Beyond cysteine: recent developments in the area of targeted covalent inhibition

2. Rapid Covalent-Probe Discovery by Electrophile-Fragment Screening

3. Fragment-Based Covalent Ligand Screening Enables Rapid Discovery of Inhibitors for the RBR E3 Ubiquitin Ligase HOIP

4. Crystallographic and electrophilic fragment screening of the SARS-CoV-2 main protease

5. Design of next-generation covalent inhibitors: Targeting residues beyond cysteine

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1. Collaborative GSK–University of Strathclyde doctoral research and training programmes: Transforming approaches to industry–academia engagement;Drug Discovery Today;2024-09

2. SuFEx Chemistry Enables Covalent Assembly of a 280-kDa 18-Subunit Pore-Forming Complex;Journal of the American Chemical Society;2024-08-27

3. Design of a covalent protein-protein interaction inhibitor of SRPKs to suppress angiogenesis and invasion of cancer cells;Communications Chemistry;2024-06-27

4. Emerging and Re-emerging Warheads for Targeted Covalent Inhibitors: An Update;Journal of Medicinal Chemistry;2024-05-07

5. Mild Strategy for the Preparation of Alkyl Sulfonyl Fluorides from Alkyl Bromides and Alcohols Using Photoredox Catalysis and Flow Chemistry;Organic Letters;2024-04-25

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