Discovery of Highly Potent and Selective Inhibitors of Neuronal Nitric Oxide Synthase by Fragment Hopping-Reference-Cited by-同舟云学术

Discovery of Highly Potent and Selective Inhibitors of Neuronal Nitric Oxide Synthase by Fragment Hopping

Published:2009-01-06 Issue:3 Volume:52 Page:779-797
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ji Haitao¹,Li Huiying¹,Martásek Pavel¹,Roman Linda J.¹,Poulos Thomas L.¹,Silverman Richard B.¹

Affiliation:

1. Department of Chemistry, Department of Biochemistry, Molecular Biology, and Cell Biology, and Center for Drug Discovery and Chemical Biology, Northwestern University, Evanston, Illinois 60208-3113, Departments of Molecular Biology and Biochemistry, Pharmaceutical Chemistry, and Chemistry, University of California, Irvine, California 92697-3900, Department of Biochemistry, The University of Texas Health Science Center, San Antonio, Texas 78384-7760, and Department of Pediatrics, First Faculty of Medicine,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm801220a

Reference73 articles.

1. Fragment-Based Drug Discovery

2. Fragment-based lead discovery

3. Fragment-based lead discovery: a chemical update

4. Recent Developments in Fragment-Based Drug Discovery

5. A decade of fragment-based drug design: strategic advances and lessons learned

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