Development of a Potent Cyclic Peptide Inhibitor of the nNOS/PSD-95 Interaction

Author:

Balboa Javier R.12,Essig Dominik J.12,Ma Sana2,Karer Nichlas2,Clemmensen Louise S.2,Pedersen Søren W.2,Joerger Andreas C.34ORCID,Knapp Stefan34ORCID,Østergaard Søren1ORCID,Strømgaard Kristian2ORCID

Affiliation:

1. Novo Nordisk A/S, Research Chemistry 3, Novo Nordisk Park, 2760 Måløv, Denmark

2. Center for Biopharmaceuticals, Department of Drug Design and Pharmacology, University of Copenhagen, Universitetsparken 2, 2100 Copenhagen, Denmark

3. Institute of Pharmaceutical Chemistry, Goethe University, Max-von-Laue Str. 9, 60438 Frankfurt am Main, Germany

4. Structural Genomics Consortium (SGC), Buchmann Institute for Molecular Life Sciences (BMLS), Max-von-Laue-Str. 15, 60438 Frankfurt am Main, Germany

Funder

Bayer

Merck KGaA

Genentech

Takeda Pharmaceutical Company

Deutsche Forschungsgemeinschaft

Pfizer

H2020 Marie Sklodowska-Curie Actions

Bristol-Myers Squibb

Genome Canada

Boehringer Ingelheim

Janssen

EUbOPEN

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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