Functionalized Scout Fragments for Site-Specific Covalent Ligand Discovery and Optimization-Reference-Cited by-同舟云学术

Functionalized Scout Fragments for Site-Specific Covalent Ligand Discovery and Optimization

Published:2021-04-05 Issue:4 Volume:7 Page:613-623
ISSN:2374-7943
Container-title:ACS Central Science
language:en
Short-container-title:ACS Cent. Sci.

Author:

Crowley Vincent M.¹^ORCID,Thielert Marvin¹,Cravatt Benjamin F.¹^ORCID

Affiliation:

1. The Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92307, United States

Funder

National Cancer Institute

National Institute of Allergy and Infectious Diseases

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acscentsci.0c01336

Reference58 articles.

1. Recent Advances in Selective and Irreversible Covalent Ligand Development and Validation

2. The promise and peril of chemical probes

3. Objective, Quantitative, Data-Driven Assessment of Chemical Probes

4. High-Throughput Kinetic Analysis for Target-Directed Covalent Ligand Discovery

5. Covalent inhibitors design and discovery

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