Covalent hits and where to find them
Author:
Funder
AstraZeneca
Publisher
Elsevier BV
Reference142 articles.
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2. The clinical KRAS(G12C) inhibitor AMG 510 drives anti-tumour immunity;Canon;Nature,2019
3. Adagrasib in non–small-cell lung cancer harboring a KRASG12C mutation;Jänne;N Engl J Med,2022
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Cited by 4 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Hit me with your best shot: Integrated hit discovery for the next generation of drug targets;Drug Discovery Today;2024-10
2. Advanced technologies for screening and identifying covalent inhibitors;TrAC Trends in Analytical Chemistry;2024-09
3. Design of a Lead-Like Cysteine-Targeting Covalent Library and the Identification of Hits to Cys55 of Bfl-1;Journal of Medicinal Chemistry;2024-06-25
4. Identification and Evaluation of Reversible Covalent Binders to Cys55 of Bfl-1 from a DNA-Encoded Chemical Library Screen;ACS Medicinal Chemistry Letters;2024-05-20
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