Recent Advances in Selective and Irreversible Covalent Ligand Development and Validation-Reference-Cited by-同舟云学术

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Recent Advances in Selective and Irreversible Covalent Ligand Development and Validation

Published:2019-11 Issue:11 Volume:26 Page:1486-1500
ISSN:2451-9456
Container-title:Cell Chemical Biology
language:en
Short-container-title:Cell Chemical Biology

Author:

Zhang Tinghu,Hatcher John M.,Teng Mingxing,Gray Nathanael S.,Kostic Milka

Funder

Linde Program in Chemical Biology

NIH

Novartis

Takeda

Astellas

Taiho

Janssen

Kinogen

Voronoi

Her2llc

Deerfield

Sanofi

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,Biochemistry

Reference86 articles.

1. Identification and characterization of an irreversible inhibitor of CDK2;Anscombe;Chem. Biol.,2015

2. The promise and peril of chemical probes;Arrowsmith;Nat. Chem. Biol.,2015

3. The pharmacological landscape and therapeutic potential of serine hydrolases;Bachovchin;Nat. Rev. Drug Discov.,2012

4. Proteome-wide covalent ligand discovery in native biological systems;Backus;Nature,2016

5. Seven year itch: pan-assay interference compounds (PAINS) in 2017—utility and limitations;Baell;ACS Chem. Biol.,2018

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1. Advanced technologies for screening and identifying covalent inhibitors;TrAC Trends in Analytical Chemistry;2024-09

2. Rationally designed BCR-ABL kinase inhibitors for improved leukemia treatment via covalent and pro-/dual-drug targeting strategies;Journal of Advanced Research;2024-09

3. Development and Application of Reversible and Irreversible Covalent Probes for Human and Mouse Cathepsin‐K Activity Detection, Revealing Nuclear Activity;Advanced Science;2024-07-05

4. Emerging and Re-emerging Warheads for Targeted Covalent Inhibitors: An Update;Journal of Medicinal Chemistry;2024-05-07

5. Histidine-Covalent Stapled Alpha-Helical Peptides Targeting hMcl-1;Journal of Medicinal Chemistry;2024-05-02

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