A Strategy Combining Differential Low-Throughput Screening and Virtual Screening (DLS-VS) Accelerating the Discovery of new Modulators for the Orphan GPR34 Receptor-Reference-Cited by-同舟云学术

A Strategy Combining Differential Low-Throughput Screening and Virtual Screening (DLS-VS) Accelerating the Discovery of new Modulators for the Orphan GPR34 Receptor

Published:2013-02 Issue:2 Volume:32 Page:213-229
ISSN:1868-1743
Container-title:Molecular Informatics
language:en
Short-container-title:Mol. Inf.

Author:

Diaz Constantino,Labit-Le Bouteiller Christine,Yvon Stéphane,Cambon-Kernëis Aimée,Roasio Annette,Jamme Marie-Françoise,Aries Amélie,Feuillerat Claude,Perret Eric,Guette Fréderique,Dieu Pierre,Miloux Brigitte,Albène Danielle,Hasel Nathalie,Kaghad Mourad,Ferran Edgardo,Lupker Jan,Ferrara Pascual

Publisher

Wiley

Subject

Organic Chemistry,Computer Science Applications,Drug Discovery,Molecular Medicine,Structural Biology

Reference85 articles.

1. Structural diversity of G protein-coupled receptors and significance for drug discovery

2. The crystallographic structure of the human adenosine A2A receptor in a high-affinity antagonist-bound state: implications for GPCR drug screening and design

3. Seven-transmembrane receptors

4. How many drug targets are there?

5. Orphan GPCRs and their ligands

Cited by 12 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Lysophosphatidylserine: A Signaling Lipid with Implications in Human Diseases;Chemical Reviews;2024-04-12

2. Structure-Based Design of a Chemical Probe Set for the 5-HT_5A Serotonin Receptor;Journal of Medicinal Chemistry;2022-02-23

3. Structure-based design of a chemical probe set for the 5-HT5A serotonin receptor;2021-12-07

4. A practical guide to large-scale docking;Nature Protocols;2021-09-24

5. Current Knowledge on the Biology of Lysophosphatidylserine as an Emerging Bioactive Lipid;Cell Biochemistry and Biophysics;2021-06-15