Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis-Reference-Cited by-同舟云学术

Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis

Published:2018-02-06 Issue:4 Volume:13 Page:321-337
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Ouvry Gilles¹^ORCID,Atrux-Tallau Nicolas¹,Bihl Franck¹,Bondu Aline¹,Bouix-Peter Claire¹,Carlavan Isabelle¹,Christin Olivier¹,Cuadrado Marie-Josée¹,Defoin-Platel Claire¹,Deret Sophie¹,Duvert Denis¹,Feret Christophe¹,Forissier Mathieu¹,Fournier Jean-François¹^ORCID,Froude David¹,Hacini-Rachinel Fériel¹,Harris Craig Steven¹,Hervouet Catherine¹,Huguet Hélène¹,Lafitte Guillaume¹,Luzy Anne-Pascale¹,Musicki Branislav¹,Orfila Danielle¹,Ozello Benjamin¹,Pascau Coralie¹,Pascau Jonathan¹,Parnet Véronique¹,Peluchon Guillaume¹,Pierre Romain¹,Piwnica David¹,Raffin Catherine¹,Rossio Patricia¹,Spiesse Delphine¹,Taquet Nathalie¹,Thoreau Etienne¹,Vatinel Rodolphe¹,Vial Emmanuel¹,Hennequin Laurent François¹

Affiliation:

1. Nestlé Skin Health R&D; 2400 Route des Colles, BP 87 06902 Sophia-Antipolis Cedex France

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Reference53 articles.

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