RORγ antagonists and inverse agonists: a patent review
Author:
Funder
Genentech
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
http://www.tandfonline.com/doi/pdf/10.1080/13543776.2017.1236918
Reference31 articles.
1. Identification of Nuclear Receptor mRNAs by RT-PCR Amplification of Conserved Zinc-Finger Motif Sequences
2. Isoform-specific amino-terminal domains dictate DNA-binding properties of ROR alpha, a novel family of orphan hormone nuclear receptors.
3. RZRs, a new family of retinoid-related orphan receptors that function as both monomers and homodimers
4. ROR-γ: The Third Member of ROR/RZR Orphan Receptor Subfamily That Is Highly Expressed in Skeletal Muscle
5. RORγt, a Novel Isoform of an Orphan Receptor, Negatively Regulates Fas Ligand Expression and IL-2 Production in T Cells
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