Changes in pH differently affect the binding properties of histamine H1 receptor antagonists
Author:
Publisher
Elsevier BV
Subject
Pharmacology
Reference36 articles.
1. Effect of race and sex on single and multiple dose pharmacokinetics of desloratadine;Affrime;Clin. Pharmacokinet.,2002
2. Biochemical characterization of desloratadine, a potent antagonist of the human histamine H1 receptor;Anthes;Eur. J. Pharmacol.,2002
3. Pharmacological differences between human and guinea pig histamine H1 receptors: Asn84 (2.61) as key residue within an additional binding pocket in the H1 receptor;Bruysters;Mol. Pharmacol.,2005
4. Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction;Cheng;Biochem. Pharmacol.,1973
5. Histamine H1 receptor antagonism by cetirizine in isolated guinea pig tissues: influence of receptor reserve and dissociation kinetics;Christophe;Eur. J. Pharmacol.,2003
Cited by 50 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Histamine/H1 receptor signaling in the parafacial region increases activity of chemosensitive neurons and respiratory activity in rats;Journal of Neurophysiology;2022-07-01
2. Assessment of receptor affinities of ophthalmic and systemic agents in dry eye disease;Current Opinion in Allergy & Clinical Immunology;2021-08-12
3. Crosstalk of physiological pH and chemical pKa under the umbrella of physiologically based pharmacokinetic modeling of drug absorption, distribution, metabolism, excretion, and toxicity;Expert Opinion on Drug Metabolism & Toxicology;2021-07-31
4. Acidification can directly affect olfaction in marine organisms;Journal of Experimental Biology;2021-07-15
5. Ocean Acidification Amplifies the Olfactory Response to 2-Phenylethylamine: Altered Cue Reception as a Mechanistic Pathway?;Journal of Chemical Ecology;2021-05-20
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3