N-Sulfonyl dipeptide nitriles as inhibitors of human cathepsin S: In silico design, synthesis and biochemical characterization
Author:
Funder
FAPESP
Publisher
Elsevier BV
Subject
Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry
Reference61 articles.
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3. Identification and pre-clinical testing of a reversible cathepsin protease inhibitor reveals anti-tumor efficacy in a pancreatic cancer model;Elie;Biochimie,2010
4. Link JO, Mossman CJ, Woo SH, Zipfel SM. Preparation of (hetero)aryltrifluoroethyl containing amino acid cyanoalkylamides as cysteine protease (cathepsin S) inhibitors. Patent US 2003-60504680. 2004.
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