Cathepsin-Targeting SARS-CoV-2 Inhibitors: Design, Synthesis, and Biological Activity

Author:

Flury Philipp1,Breidenbach Julian2,Krüger Nadine3,Voget Rabea2,Schäkel Laura2,Si Yaoyao2,Krasniqi Vesa2,Calistri Sara1,Olfert Matthias4,Sylvester Katharina2,Rocha Cheila3,Ditzinger Raphael1,Rasch Alexander1,Pöhlmann Stefan34,Kronenberger Thales156,Poso Antti15ORCID,Rox Katharina78,Laufer Stefan A.1ORCID,Müller Christa E.2ORCID,Gütschow Michael2ORCID,Pillaiyar Thanigaimalai1ORCID

Affiliation:

1. Institute of Pharmacy, Pharmaceutical/Medicinal Chemistry and Tübingen Center for Academic Drug Discovery, Eberhard Karls University Tübingen, Auf der Morgenstelle 8, Tübingen 72076, Germany

2. PharmaCenter Bonn, Pharmaceutical Institute, Pharmaceutical & Medicinal Chemistry, University of Bonn, An der Immenburg 4, Bonn 53121, Germany

3. Infection Biology Unit, German Primate Center, Leibniz Institute for Primate Research Göttingen, Kellnerweg 4, Göttingen 37077, Germany

4. Faculty of Biology and Psychology, University Göttingen, Göttingen 37073, Germany

5. Faculty of Health Sciences, School of Pharmacy, University of Eastern Finland, Kuopio 70211, Finland

6. Excellence Cluster “Controlling Microbes to Fight Infections” (CMFI), Tübingen 72076, Germany

7. Department of Chemical Biology, Helmholtz Centre for Infection Research (HZI), Braunschweig 38124, Germany

8. Partner Site Hannover-Braunschweig, German Center for Infection Research (DZIF), Braunschweig 38124, Germany

Publisher

American Chemical Society (ACS)

Subject

Pharmacology (medical),Pharmacology

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3