Identification and pre-clinical testing of a reversible cathepsin protease inhibitor reveals anti-tumor efficacy in a pancreatic cancer model

Author:

Elie Benelita Tina,Gocheva Vasilena,Shree Tanaya,Dalrymple Stacie A.,Holsinger Leslie J.,Joyce Johanna A.

Funder

National Cancer Institute

NIH Cancer Center Support grant

Geoffrey Beene Foundation

Publisher

Elsevier BV

Subject

General Medicine,Biochemistry

Reference48 articles.

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3. Tumour microenvironment - opinion: validating matrix metalloproteinases as drug targets and anti-targets for cancer therapy;Overall;Nat. Rev. Cancer,2006

4. Cysteine cathepsin proteases as pharmacological targets in cancer;Palermo;Trends Pharmacol. Sci.,2008

5. The urokinase plasminogen activator system: a target for anti-cancer therapy;Ulisse;Curr. Cancer Drug Targets,2009

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