A Simple HPLC Assay for Proguanil and Its Active Metabolite Cycloguanil: Application to Oxidation Phenotyping
Author:
Affiliation:
1. a School of Pharmacy, Univeristy of Otago , P.O. Box 913, Dunedin , New Zealand
Publisher
Informa UK Limited
Subject
Molecular Medicine
Link
https://www.tandfonline.com/doi/pdf/10.1080/10826079508013747
Reference12 articles.
1. Inter-subject variability in the metabolism of proguanil to the active metabolite cycloguanil in man.
2. The pharmacokinetics and activation of proguanil in man: consequences of variability in drug metabolism.
3. The activation of the biguanide antimalarial proguanil co-segregates with the mephenytoin oxidation polymorphism-a panel study.
4. The multiple dose pharmacokinetics of proguanil.
5. Variability in the metabolism of proguanil to the active metabolite cycloguanil in healthy Kenyan adults
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2. Bioanalysis of antimalarials using liquid chromatography;TrAC Trends in Analytical Chemistry;2013-01
3. Alternative LC–MS–MS Method for Simultaneous Determination of Proguanil, Its Active Metabolite in Human Plasma and Application to a Bioequivalence Study;Chromatographia;2009-07-31
4. Genetic polymorphism of debrisoquine (CYP2D6) and proguanil (CYP2C19) in South Pacific Polynesian populations;European Journal of Clinical Pharmacology;1998-08-17
5. Improved Validated Assay for the Determination of Proguanil and Its Metabolites in Plasma, Whole Blood, and Urine Using Solid-Phase Extraction and High-Performance Liquid Chromatography;Therapeutic Drug Monitoring;1998-06
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