Fluorescence-Based, High-Throughput Assays for μ-Opioid Receptor Activation Using a Membrane Potential-Sensitive Dye-Reference-Cited by-同舟云学术

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Fluorescence-Based, High-Throughput Assays for μ-Opioid Receptor Activation Using a Membrane Potential-Sensitive Dye

Published:2014-09-15 Issue: Volume: Page:177-185
ISSN:1064-3745
Container-title:Methods in Molecular Biology
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Author:

Knapman Alisa,Connor Mark

Publisher

Springer New York

Link

http://link.springer.com/content/pdf/10.1007/978-1-4939-1708-2_14

Reference16 articles.

1. Matthes HWD, Maldonado R, Simonin F et al (1996) Loss of morphine-induced analgesia, reward effect and withdrawal symptoms in mice lacking the μ-opioid-receptor gene. Nature 383:819–823

2. Kenakin T, Miller LJ (2010) Seven transmembrane receptors as shapeshifting proteins: the impact of allosteric modulation and functional selectivity on new drug discovery. Pharmacol Rev 62:265–304

3. Pinyero G, Archer-Lahlou E (2007) Ligand-specific receptor states: implications for opiate receptor signaling and regulation. Cell Signal 19:8–19

4. DeWire SM, Yamashita DS, Rominger DH et al (2013) A G protein-biased ligand at the μ-opioid receptor is potently analgesic with reduced gastrointestinal and respiratory dysfunction compared with morphine. J Pharmacol Exp Ther 344:708–717

5. Kenakin T, Christopoulos A (2013) Signalling bias in new drug discovery: detection, quantification and therapeutic impact. Nat Rev Drug Discov 12:205–216

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