Discovery of fragments inducing conformational effects in dynamic proteins using a second-harmonic generation biosensor-Reference-Cited by-同舟云学术

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Discovery of fragments inducing conformational effects in dynamic proteins using a second-harmonic generation biosensor

Published:2021 Issue:13 Volume:11 Page:7527-7537
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

FitzGerald Edward A.¹²³⁴⁵^ORCID,Butko Margaret T.⁶⁷⁸,Boronat Pierre⁹¹⁰¹¹¹²¹³,Cederfelt Daniela¹²³⁴,Abramsson Mia¹²³⁴^ORCID,Ludviksdottir Hildur¹²³⁴,van Muijlwijk-Koezen Jacqueline E.⁹¹⁰¹¹¹²¹³,de Esch Iwan J. P.⁹¹⁰¹¹¹²¹³,Dobritzsch Doreen¹²³⁴,Young Tracy⁶⁷⁸,Danielson U. Helena¹²³⁴¹⁴^ORCID

Affiliation:

1. Department of Chemistry – BMC

2. Uppsala University

3. Uppsala

4. Sweden

5. Beactica Therapeutics

6. Biodesy, Inc.

7. South San Francisco

8. USA

9. Amsterdam Institute of Molecular and Life Sciences (AIMMS)

10. Division of Medicinal Chemistry

11. Faculty of Science

12. Vrije Universiteit Amsterdam

13. HZ Amsterdam

14. Science for Life Laboratory

Abstract

Fragments inducing conformational changes identified at a dynamic region of AChBP.

Funder

H2020 Marie Skłodowska-Curie Actions

Science for Life Laboratory

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/RA/D0RA09844B

Reference36 articles.

1. On the nature of allosteric transitions: A plausible model

2. Structures of Aplysia AChBP complexes with nicotinic agonists and antagonists reveal distinctive binding interfaces and conformations

3. Loop C and the mechanism of acetylcholine receptor–channel gating

4. Design, Synthesis, and Structure–Activity Relationships of Highly Potent 5-HT3 Receptor Ligands

5. Use of Acetylcholine Binding Protein in the Search for Novel α7 Nicotinic Receptor Ligands. In Silico Docking, Pharmacological Screening, and X-ray Analysis

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