Design, Synthesis, and Structure–Activity Relationships of Highly Potent 5-HT3 Receptor Ligands-Reference-Cited by-同舟云学术

Design, Synthesis, and Structure–Activity Relationships of Highly Potent 5-HT3 Receptor Ligands

Published:2012-10-12 Issue:20 Volume:55 Page:8603-8614
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Verheij Mark H. P.¹,Thompson Andrew J.²,van Muijlwijk-Koezen Jacqueline E.¹,Lummis Sarah C. R.²,Leurs Rob¹,de Esch Iwan J. P.¹

Affiliation:

1. Leiden/Amsterdam Center of Drug Research (LACDR), Amsterdam Institute for Molecules Medicines and Systems (AIMMS), Division of Medicinal Chemistry, Faculty of Sciences, VU University Amsterdam, Amsterdam, The Netherlands.

2. Department of Biochemistry, University of Cambridge, Cambridge, United Kingdom

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300801u

Reference50 articles.

1. A Review of Granisetron, 5-Hydroxytryptamine3 Receptor Antagonists, and Other Antiemetics

2. Targeting the 5-HT3 receptor in the treatment of irritable bowel syndrome

3. Review: The auspicious role of the 5-HT3 receptor in depression: a probable neuronal target?

4. The 5-HT3receptor as a therapeutic target

5. Primary Structure And Functional Expression of the 5HT 3 Receptor, A Serotonin-gated Ion Channel

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