Brønsted acid-promoted ring-opening and annulation of thioamides and 2<i>H</i>-azirines to synthesize 2,4,5-trisubstituted thiazoles-Reference-Cited by-同舟云学术

Brønsted acid-promoted ring-opening and annulation of thioamides and 2H-azirines to synthesize 2,4,5-trisubstituted thiazoles

Published:2023 Issue:27 Volume:21 Page:5532-5536
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Wang Meng¹,Ma Jingyi¹,Wang Hesong¹,Hu Fangpeng¹,Sun Bo¹,Tan Taiyan¹,Li Minglang¹,Huang Guosheng¹^ORCID

Affiliation:

1. State Key Laboratory of Applied Organic Chemistry, Key Laboratory of Nonferrous Metal Chemistry and Resources Utilization of Gansu Province, Department of Chemistry, Lanzhou University, Lanzhou 730000, China

Abstract

We have developed a metal-free synthesis method of 2,4,5-trisubstituted thiazoles by the formation of C–S and C–N bonds.It is a green and efficient way with a broad substrate scope. And this protocol features mild conditions and simple operation.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2023/OB/D3OB00245D

Reference49 articles.

1. Highly Flexible π-Expanded Cyclooctatetraenes: Cyclic Thiazole Tetramers with Head-to-Tail Connection

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4. Mutations of β-tubulin codon 198 or 200 indicate thiabendazole resistance among isolates of Penicillium digitatum collected from citrus in Taiwan

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