Hypervalent iodine(<scp>iii</scp>) promoted tandem reaction of <i>o</i>-fluoroanilines with formamides to construct 2-aminobenzoxazoles-Reference-Cited by-同舟云学术

Hypervalent iodine(iii) promoted tandem reaction of o-fluoroanilines with formamides to construct 2-aminobenzoxazoles

Published:2022 Issue:9 Volume:9 Page:2412-2417
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Long Lipeng¹,Wang Jieyan¹,Li Xin¹,Peng ShunFeng¹,Qiao Liang¹,Luo Guotian¹,Chen Zhengwang¹^ORCID

Affiliation:

1. Key Laboratory of Organo-pharmaceutical Chemistry of Jiangxi Province, Gannan Normal University, Ganzhou, 341000, China

Abstract

A novel catalyst-free hypervalent iodine(iii)-promoted tandem nucleophilic addition/aromatic nucleophilic substitution reaction of o-fluoroanilines with formamides toward 2-aminobenzoxazoles.

Funder

Natural Science Foundation of Jiangxi Province

Bureau of Science and Technology of Ganzhou Municipality

Education Department of Jiangxi Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2022/QO/D2QO00049K

Reference43 articles.

1. Design, Synthesis, and Evaluation of Orally Active Benzimidazoles and Benzoxazoles as Vascular Endothelial Growth Factor-2 Receptor Tyrosine Kinase Inhibitors

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3. Identification of a series of benzoxazoles as potent 5-HT6 ligands

4. Discovery of the Dual Orexin Receptor Antagonist [(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone (MK-4305) for the Treatment of Insomnia

5. Orally Active Benzoxazole Derivative as 5-HT3 Receptor Partial Agonist for Treatment of Diarrhea-Predominant Irritable Bowel Syndrome

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