Synthesis of polysubstituted 4-aminopyrazoles and 4-hydroxypyrazoles from vinyl azides and hydrazines
Author:
Affiliation:
1. Zhejiang Province Key Laboratory of Anti-Cancer Drug Research
2. College of Pharmaceutical Science
3. Zhejiang University
4. Hangzhou 310058
5. P. R. China
Abstract
A simple and direct synthesis of polysubstituted 4-aminopyrazoles and 4-hydroxypyrazoles from vinyl azides and hydrazines.
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemical Engineering,General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA04371A
Reference25 articles.
1. Identification of N-(4-Piperidinyl)-4-(2,6-dichlorobenzoylamino)-1H-pyrazole-3-carboxamide (AT7519), a Novel Cyclin Dependent Kinase Inhibitor Using Fragment-Based X-Ray Crystallography and Structure Based Drug Design
2. Discovery and Development of Pyrazole-Scaffold Hsp90 Inhibitors
3. Discovery of Highly Potent, Selective, and Brain-Penetrant Aminopyrazole Leucine-Rich Repeat Kinase 2 (LRRK2) Small Molecule Inhibitors
4. Property- and Structure-Guided Discovery of a Tetrahydroindazole Series of Interleukin-2 Inducible T-Cell Kinase Inhibitors
5. Discovery of Potent and Selective Pyrazolopyrimidine Janus Kinase 2 Inhibitors
Cited by 12 articles. 订阅此论文施引文献 订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献
1. Recent Advances in the Use of α‐Azidochalcones in Heterocycle Synthesis;Advanced Synthesis & Catalysis;2024-06-16
2. Discovery of 4-hydroxyl pyrazole derivatives as potent ferroptosis inhibitors;European Journal of Medicinal Chemistry;2024-01
3. Recent Advances on α ‐Azidoketones and Esters in the Synthesis of N ‐Heterocycles;Asian Journal of Organic Chemistry;2022-06-24
4. Recent advances in pyrazole synthesis employing diazo compounds and synthetic analogues;Organic & Biomolecular Chemistry;2022
5. Vinylazides: versatile synthons and magical precursors for the construction of N-heterocycles;Molecular Diversity;2020-05-30
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3