Three successive and regiocontroled palladium cross-coupling reactions to easily synthesize novel series of 2,4,6-tris(het)aryl pyrido[1′,2′:1,5]pyrazolo[3,4-d]pyrimidines-Reference-Cited by-同舟云学术

Three successive and regiocontroled palladium cross-coupling reactions to easily synthesize novel series of 2,4,6-tris(het)aryl pyrido[1′,2′:1,5]pyrazolo[3,4-d]pyrimidines

Published:2018 Issue:2 Volume:8 Page:732-741
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Belaroussi R.¹²³⁴⁵,Ejjoummany A.¹²³⁴⁵,El Hakmaoui A.⁶⁷⁸⁹¹⁰,Akssira M.⁶⁷⁸⁹¹⁰,Guillaumet G.¹²³⁴⁵^ORCID,Routier S.¹²³⁴⁵^ORCID

Affiliation:

1. Univ Orleans

2. CNRS

3. Institut de Chimie Organique et Analytique

4. 45067 Orléans Cedex 2

5. France

6. Laboratoire de Chimie Physique et Chimie Bioorganique

7. FST Mohammedia

8. Université Hassan II de Casablanca

9. 28800 Mohammedia

10. Morocco

Abstract

The first access to tris(het)arylated pyrido[1′,2′:1,5]pyrazolo[3,4-d]pyrimidine derivatives is reported.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/RA/C7RA12246B

Reference33 articles.

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3. Pyrazolo[1,5-a]pyridines as p38 Kinase Inhibitors

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5. Synthesis of a Novel Series of Tricyclic Dihydrofuran Derivatives: Discovery of 8,9-Dihydrofuro[3,2-c]pyrazolo[1,5-a]pyridines as Melatonin Receptor (MT1/MT2) Ligands

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