Discovery of 6-Oxo-3-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1(6H)-pyridazinebutanoic Acid (FK 838): A Novel Non-Xanthine Adenosine A1 Receptor Antagonist with Potent Diuretic Activity-Reference-Cited by-同舟云学术

Discovery of 6-Oxo-3-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1(6H)-pyridazinebutanoic Acid (FK 838): A Novel Non-Xanthine Adenosine A1 Receptor Antagonist with Potent Diuretic Activity

Published:1999-02-20 Issue:5 Volume:42 Page:779-783
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Akahane Atsushi¹,Katayama Hirohito¹,Mitsunaga Takafumi¹,Kato Takeshi¹,Kinoshita Takayoshi¹,Kita Yasuhiro¹,Kusunoki Takahiro¹,Terai Takao¹,Yoshida Keizo¹,Shiokawa Youichi¹

Affiliation:

1. Medicinal Chemistry Research Laboratories, Fujisawa Pharmaceutical Company, Ltd., 1-6, 2-chome, Kashima, Yodogawa-ku, Osaka 532-8514, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm980671w

Reference25 articles.

1. Adenosine receptor subtypes

2. A1-Adenosine receptor antagonists

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