In situ generation and trapping of thioimidates: an intermolecular tandem reaction to 4-acylimino-4H-3,1-benzothiazines-Reference-Cited by-同舟云学术

In situ generation and trapping of thioimidates: an intermolecular tandem reaction to 4-acylimino-4H-3,1-benzothiazines

Published:2016 Issue:19 Volume:6 Page:15430-15440
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Steinebach Christian¹²³⁴⁵,Schulz-Fincke Anna-Christina¹²³⁴⁵,Schnakenburg Gregor⁶³⁴⁵,Gütschow Michael¹²³⁴⁵

Affiliation:

1. Pharmaceutical Institute

2. Pharmaceutical Chemistry I

3. University of Bonn

4. D-53121 Bonn

5. Germany

6. Institute of Inorganic Chemistry

Abstract

The proton-catalyzed transformation of 2-thioureidobenzonitriles in the presence of acyl donors provides a convenient one-step entry to 4-acylimino-4H-3,1-benzothiazines.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/RA/C6RA00196C

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