Thiosulfonylation of alkenes with the insertion of sulfur dioxide under non-metallic conditions-Reference-Cited by-同舟云学术

Thiosulfonylation of alkenes with the insertion of sulfur dioxide under non-metallic conditions

Published:2018 Issue:20 Volume:5 Page:2940-2944
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

He Fu-Sheng¹²³⁴,Wu Youqian¹²³⁴,Zhang Jun⁵⁶⁷⁴,Xia Hongguang¹²³⁴,Wu Jie⁵⁶⁷⁴⁸^ORCID

Affiliation:

1. Department of Biochemistry & Research Center of Clinical Pharmacy of The First Affiliated Hospital

2. Zhejiang University School of Medicine

3. Hangzhou 310058

4. China

5. Department of Chemistry

6. Fudan University

7. Shanghai 200438

8. State Key Laboratory of Organometallic Chemistry

Abstract

A three-component reaction of 1-(2-allylaryl)thioureas, sulfur dioxide, and aryldiazonium tetrafluoroborates under mild conditions is realized, leading to sulfonated [3,1]-benzothiazepines in good yields. High efficiency is observed for this non-metallic transformation.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/QO/C8QO00824H

Reference125 articles.

1. 1,5-Benzothiazepine, a versatile pharmacophore: A review

2. L-Type Calcium Channel Blockers: From Diltiazem to 1,2,4-Oxadiazol-5-ones via Thiazinooxadiazol-3-one Derivatives

3. Torn from the Headlines: AstraZeneca Fined For Illegal Marketing of SEROQUEL