Diversified syntheses of multifunctionalized thiazole derivatives via regioselective and programmed C

Diversified syntheses of multifunctionalized thiazole derivatives via regioselective and programmed C–H activation

Published:2015 Issue:22 Volume:51 Page:4599-4602
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Liu Xiang-Wei¹²³⁴⁵,Shi Jiang-Ling⁶⁷⁵,Wei Jiang-Bo¹²³⁴⁵,Yang Chao⁸⁹⁵,Yan Jia-Xuan¹²³⁴⁵,Peng Kun¹⁰¹¹¹²¹³⁵,Dai Le¹⁰¹¹¹²¹³⁵,Li Chen-Guang¹⁰¹¹¹²¹³⁵,Wang Bi-Qin⁶⁷⁵,Shi Zhang-Jie¹²³⁴⁵

Affiliation:

1. Beijing National Laboratory of Molecular Sciences (BNLMS) and Key Laboratory of Bioorganic Chemistry and Molecular Engineering of Ministry of Education

2. College of Chemistry

3. Peking University

4. Beijing 100871

5. China

6. College of Chemistry and Material Chemistry

7. Sichuan Normal University

8. Shenzhen Graduate School of Peking University

9. Shenzhen 518055

10. DSM nutritional products

11. DSM nutrition center

12. DSM (China) limited

13. Shanghai

Abstract

The direct construction of 5-alkenylated thiazole derivatives from 2-/4-substituted thiazole derivatives or challenging thiazole via palladium-catalyzed regioselective 5-alkenylation has been realized.

Funder

Ministry of Science and Technology

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2015/CC/C4CC10419F

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5. Sequential C–H Functionalization Reactions for the Enantioselective Synthesis of Highly Functionalized 2,3-Dihydrobenzofurans

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