Diversified facile synthesis of benzimidazoles, quinazolin-4(3H)-ones and 1,4-benzodiazepine-2,5-diones via palladium-catalyzed transfer hydrogenation/condensation cascade of nitro arenes under microwave irradiation-Reference-Cited by-同舟云学术

Diversified facile synthesis of benzimidazoles, quinazolin-4(3H)-ones and 1,4-benzodiazepine-2,5-diones via palladium-catalyzed transfer hydrogenation/condensation cascade of nitro arenes under microwave irradiation

Published:2015 Issue:15 Volume:5 Page:11132-11135
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Zhu Kaicheng¹²³⁴⁵,Hao Jian-Hong¹²³⁴⁵,Zhang Cheng-Pan¹²³⁴⁵,Zhang Jiajun¹²³⁴⁵,Feng Yiqing¹²³⁴⁵,Qin Hua-Li¹²³⁴⁵

Affiliation:

1. School of Chemistry

2. Chemical Engineering and Life Science

3. Wuhan University of Technology

4. Wuhan

5. P. R. China

Abstract

An efficient methodology for diversified preparation of benzimidazole, quinazolin-4(3H)-ones and 1,4-benzodiazepine-2,5-diones is established using a Pd-CTH/condensation cascade of nitro arenes in a TEA–formic acid mixture under microwave irradiation.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/RA/C4RA15765F

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2. Studies on Quinazolines. 11. Intramolecular Imidate-Amide Rearrangement of 2-Substituted 4-(ω-Chloroalkoxy)quinazoline Derivatives. 1,3 -O → N Shift of Chloroalkyl Groups via Cyclic 1,3-Azaoxonium Intermediates

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