A [two-step/one week] synthesis of C-functionalized homocyclens and cyclams. Application to the preparation of conjugable BCAs without chelating properties alteration-Reference-Cited by-同舟云学术

A [two-step/one week] synthesis of C-functionalized homocyclens and cyclams. Application to the preparation of conjugable BCAs without chelating properties alteration

Published:2015 Issue:104 Volume:5 Page:85898-85910
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Camus Nathalie¹²³⁴,Halime Zakaria¹²³⁴,le Bris Nathalie¹²³⁴,Bernard Hélène¹²³⁴,Beyler Maryline¹²³⁴,Platas-Iglesias Carlos⁵⁶⁷⁸⁹,Tripier Raphaël¹²³⁴

Affiliation:

1. Université de Brest

2. UMR-CNRS 6521/SFR148 ScInBioS UFR Sciences et Techniques

3. 29238 Brest

4. France

5. Grupo QUICOOR

6. Centro de Investigaciones Científicas Avanzadas (CICA) and Departamento de Química Fundamental

7. Universidade da Coruña

8. Campus da Zapateira

9. 15008 A Coruña

Abstract

An efficient synthesis ofC-functionalized azamacrocycles is presented together with a coordination study showing the week influence of the added appended group.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA17133D

Reference49 articles.

1. Thermodynamic and Kinetic Data for Macrocycle Interaction with Cations, Anions, and Neutral Molecules

2. Metal complexes of cyclen and cyclam derivatives useful for medical applications: a discussion based on thermodynamic stability constants and structural data

3. Biomedical applications of macrocyclic ligand complexes

4. Coordinating Radiometals of Copper, Gallium, Indium, Yttrium, and Zirconium for PET and SPECT Imaging of Disease

5. Matching chelators to radiometals for radiopharmaceuticals

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