Copper(i)-catalyzed asymmetric [3 + 3] annulation involving aziridines to construct tetrahydro-β-carbolines-Reference-Cited by-同舟云学术

Copper(i)-catalyzed asymmetric [3 + 3] annulation involving aziridines to construct tetrahydro-β-carbolines

Published:2020 Issue:21 Volume:7 Page:3393-3398
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Ye Chao¹²³⁴⁵,Yang Wu-Lin⁶⁷⁸⁵¹^ORCID,Zhai Yufei⁶⁷⁸⁵,Deng Hua¹²³⁴⁵,Luo Xiaoyan¹²³⁴⁵^ORCID,Kai Guoyin⁶⁷⁸⁵,Deng Wei-Ping⁶⁷⁸⁵¹^ORCID

Affiliation:

1. Shanghai Key Laboratory of New Drug Design

2. School of Pharmacy

3. East China University of Science and Technology

4. Shanghai 200237

5. China

6. College of Pharmacy

7. Zhejiang Chinese Medical University

8. Hangzhou 310053

Abstract

A copper-catalyzed asymmetric [3 + 3] annulation of 2-vinylindoles with 2-aryl aziridines has been described, providing direct access to enantioenriched tetrahydro-β-carbolines.

Funder

National Natural Science Foundation of China

Zhejiang Provincial Program for the Cultivation of High-Level Innovative Health Talents

Zhejiang Chinese Medical University

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/QO/D0QO00742K

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