Microwave-assisted synthesis of 3-aminobenzo[b]thiophene scaffolds for the preparation of kinase inhibitors
Author:
Affiliation:
1. Department of Chemistry
2. School of Life Sciences
3. University of Sussex
4. Brighton, East Sussex
5. UK
6. WestCHEM
7. Department of Pure and Applied Chemistry
8. University of Strathclyde
9. Glasgow
Abstract
Microwave-assisted synthesis of 3-aminobenzo[b]thiophenes has been applied to 3 kinase inhibitor scaffolds.
Funder
Engineering and Physical Sciences Research Council
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2015/OB/C5OB00819K
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4. A new anti-tubulin agent containing the benzo[b]thiophene ring system
5. Synthesis and Biological Evaluation of 2- and 3-Aminobenzo[b]thiophene Derivatives as Antimitotic Agents and Inhibitors of Tubulin Polymerization
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