Rhodium-catalyzed iminoiodane-mediated oxyamidation studies of 5-vinyluracil derivatives using aryl and alkyl sulfamates-Reference-Cited by-同舟云学术

Rhodium-catalyzed iminoiodane-mediated oxyamidation studies of 5-vinyluracil derivatives using aryl and alkyl sulfamates

Published:2020 Issue:37 Volume:18 Page:7414-7424
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Wang Zhaoxin¹²³⁴⁵,Jin Zongxin¹²³⁴⁵,Zhong Quanxing¹²³⁴⁵,Zhang Yinan¹²³⁴⁵,Wu Yan¹²³⁴⁵,Ma Yujiao¹²³⁴⁵,Sun Hua¹²³⁴⁵,Yu Peng¹²³⁴⁵,Dodd Robert H.¹²³⁴⁵^ORCID

Affiliation:

1. China International Science and Technology Cooperation Base of Food Nutrition/Safety and Medicinal Chemistry

2. College of Biotechnology

3. Tianjin University of Science & Technology

4. Tianjin

5. China

Abstract

Highly functionalized uracil derivatives were synthesized by regioselective intermolecular 1,2-oxyamidation of 5-vinyluracils. Selected products displayed significant α-glucosidase inhibition.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Tianjin City

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/OB/D0OB01548B

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