Mechanism of intracellular allosteric β2AR antagonist revealed by X-ray crystal structure-Reference-Cited by-同舟云学术

Mechanism of intracellular allosteric β2AR antagonist revealed by X-ray crystal structure

Published:2017-08 Issue:7668 Volume:548 Page:480-484
ISSN:0028-0836
Container-title:Nature
language:en
Short-container-title:Nature

Author:

Liu Xiangyu,Ahn Seungkirl,Kahsai Alem W.,Meng Kai-Cheng,Latorraca Naomi R.,Pani Biswaranjan,Venkatakrishnan A. J.,Masoudi Ali,Weis William I.,Dror Ron O.,Chen Xin,Lefkowitz Robert J.,Kobilka Brian K.

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/nature23652.pdf

Reference40 articles.

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3. Zheng, Y. et al. Structure of CC chemokine receptor 2 with orthosteric and allosteric antagonists. Nature 540, 458–461 (2016)

4. Oswald, C. et al. Intracellular allosteric antagonism of the CCR9 receptor. Nature 540, 462–465 (2016)

5. Jazayeri, A. et al. Extra-helical binding site of a glucagon receptor antagonist. Nature 533, 274–277 (2016)

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