Structure of CC chemokine receptor 2 with orthosteric and allosteric antagonists-Reference-Cited by-同舟云学术

Structure of CC chemokine receptor 2 with orthosteric and allosteric antagonists

Published:2016-12-07 Issue:7633 Volume:540 Page:458-461
ISSN:0028-0836
Container-title:Nature
language:en
Short-container-title:Nature

Author:

Zheng Yi,Qin Ling,Zacarías Natalia V. Ortiz,de Vries Henk,Han Gye Won,Gustavsson Martin,Dabros Marta,Zhao Chunxia,Cherney Robert J.,Carter Percy,Stamos Dean,Abagyan Ruben,Cherezov Vadim,Stevens Raymond C.,IJzerman Adriaan P.,Heitman Laura H.,Tebben Andrew,Kufareva Irina,Handel Tracy M.

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/nature20605.pdf

Reference42 articles.

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3. Lim, S. Y., Yuzhalin, A. E., Gordon-Weeks, A. N. & Muschel, R. J. Targeting the CCL2-CCR2 signaling axis in cancer metastasis. Oncotarget 7, 28697–28710 (2016)

4. Solari, R., Pease, J. E. & Begg, M. “Chemokine receptors as therapeutic targets: why aren’t there more drugs?”. Eur. J. Pharmacol. 746, 363–367 (2015)

5. Cooke, R. M., Brown, A. J., Marshall, F. H. & Mason, J. S. Structures of G protein-coupled receptors reveal new opportunities for drug discovery. Drug Discov. Today 20, 1355–1364 (2015)

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