Protein-observed 19F-NMR for fragment screening, affinity quantification and druggability assessment-Reference-Cited by-同舟云学术

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Protein-observed 19F-NMR for fragment screening, affinity quantification and druggability assessment

Published:2016-07-14 Issue:8 Volume:11 Page:1414-1427
ISSN:1754-2189
Container-title:Nature Protocols
language:en
Short-container-title:Nat Protoc

Author:

Gee Clifford T,Arntson Keith E,Urick Andrew K,Mishra Neeraj K,Hawk Laura M L,Wisniewski Andrea J,Pomerantz William C K

Publisher

Springer Science and Business Media LLC

Subject

General Biochemistry, Genetics and Molecular Biology

Link

http://www.nature.com/articles/nprot.2016.079.pdf

Reference60 articles.

1. Lepre, C.A. Practical aspects of NMR-based fragment screening. Methods Enzymol. 493, 219–239 (2011).

2. Dalvit, C. et al. A General NMR method for rapid, efficient, and reliable biochemical screening. J. Am. Chem. Soc. 125, 14620–14625 (2003).

3. Fielding, L. NMR methods for the determination of protein-ligand dissociation constants. Curr. Top. Med. Chem. 3, 39–53 (2003).

4. Williamson, M.P. Using chemical shift perturbation to characterise ligand binding. Prog. Nucl. Magn. Reson. Spectrosc. 73, 1–16 (2013).

5. Tanaka, D. et al. A Practical use of ligand efficiency indices out of the fragment-based approach: ligand efficiency-guided lead identification of soluble epoxide hydrolase inhibitors. J. Med. Chem. 54, 851–857 (2010).

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