Dynamic ligand binding dictates partial agonism at a G protein–coupled receptor-Reference-Cited by-同舟云学术

Dynamic ligand binding dictates partial agonism at a G protein–coupled receptor

Published:2013-11-10 Issue:1 Volume:10 Page:18-20
ISSN:1552-4450
Container-title:Nature Chemical Biology
language:en
Short-container-title:Nat Chem Biol

Author:

Bock Andreas,Chirinda Brian,Krebs Fabian,Messerer Regina,Bätz Julia,Muth Mathias,Dallanoce Clelia,Klingenthal Dominika,Tränkle Christian,Hoffmann Carsten,De Amici Marco,Holzgrabe Ulrike,Kostenis Evi,Mohr Klaus

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Molecular Biology

Link

http://www.nature.com/articles/nchembio.1384.pdf

Reference31 articles.

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3. Kenakin, T. Nat. Rev. Drug Discov. 1, 103–110 (2002).

4. Kenakin, T. & Christopoulos, A. Nat. Rev. Drug Discov. 12, 205–216 (2013).

5. Rosenbaum, D.M., Rasmussen, S.G.F. & Kobilka, B.K. Nature 459, 356–363 (2009).

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