Development of Blood–Brain Barrier Permeable Nitrocatechol-Based Catechol O-Methyltransferase Inhibitors with Reduced Potential for Hepatotoxicity

Author:

Silva Tiago1,Mohamed Tarek2,Shakeri Arash2,Rao Praveen P. N.2,Martínez-González Loreto3,Pérez Daniel I.3,Martínez Ana3,Valente Maria João4,Garrido Jorge5,Uriarte Eugenio6,Serrão Paula78,Soares-da-Silva Patrício78,Remião Fernando4,Borges Fernanda1

Affiliation:

1. CIQ/Department of Chemistry and Biochemistry, Faculty of Sciences, University of Porto, Rua do Campo Alegre s/n, 4169-007 Porto, Portugal

2. School of Pharmacy, Health Sciences Campus, University of Waterloo, 200 University Avenue West, Waterloo, Ontario N2L 3G1, Canada

3. Centro de Investigaciónes Biológicas, CSIC, C/Ramiro de Maeztu, 28040 Madrid, Spain

4. Laboratory of Toxicology, Department of Biological Sciences, Faculty of Pharmacy, UCIBIO-REQUIMTE, Rua de Jorge Viterbo Ferreira, 4050-313 Porto, Portugal

5. Departamento de Engenharia Química, Instituto Superior de Engenharia do Porto (ISEP), Instituto Politécnico Porto, 4200-072 Porto, Portugal

6. Department of Organic Chemistry, Faculty of Pharmacy, University of Santiago de Compostela, 15782 Santiago de Compostela, Spain

7. Department of Pharmacology and Therapeutics, Faculty of Medicine, University of Porto, 4200-319 Porto, Portugal

8. MedInUP—Center for Drug Discovery and Innovative Medicines, University of Porto, 4200-319, Porto, Portugal

Funder

Ontario Mental Health Foundation

Canada Foundation for Innovation

European Cooperation in Science and Technology

Natural Sciences and Engineering Research Council of Canada

Fundação para a Ciência e a Tecnologia

Ontario Ministry of Research and Innovation

Ontario Research Fund

European Regional Development Fund

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3